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MedKoo Cat#: 573130 | Name: Amezinium

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Amezinium is a sympathomimetic drug used for the treatment of low blood pressure. It has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake.

Chemical Structure

Amezinium
Amezinium
CAS#41658-78-0

Theoretical Analysis

MedKoo Cat#: 573130

Name: Amezinium

CAS#: 41658-78-0

Chemical Formula: C11H12N3O

Exact Mass: 202.0975

Molecular Weight: 202.24

Elemental Analysis: C, 65.33; H, 5.98; N, 20.78; O, 7.91

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Amezinium; BRN 4141517
IUPAC/Chemical Name
4-Amino-6-methoxy-1-phenylpyridazinium
InChi Key
VXROHTDSRBRJLN-UHFFFAOYSA-O
InChi Code
1S/C11H11N3O/c1-15-11-7-9(12)8-13-14(11)10-5-3-2-4-6-10/h2-8,12H,1H3/p+1
SMILES Code
COc1cc(cn[n+]1c2ccccc2)N
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 202.24 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Shimizu I, Ishii D, Kawashima K, Oka M, Hosoki K. Pharmacological effect of amezinium on urethra and bladder of rabbits. Int Urogynecol J Pelvic Floor Dysfunct. 2001;12(3):170-7. PubMed PMID: 11451005. 2: Belz GG, Aust PE, Belz G, Appel E, Palm D. Sympathomimetic effects of amezinium on the cardiovascular system and plasma catecholamines in man. Eur J Clin Pharmacol. 1982;23(1):15-20. PubMed PMID: 7128668. 3: Traut M, Brode E, Neumann B, Kummer H. Pharmacokinetics of amezinium in rat and dog. Arzneimittelforschung. 1981;31(9a):1594-604. PubMed PMID: 7197974. 4: Lenke D, Gries J, Kretzschmar R. Pharmacology of amezinium, a novel antihypotensive drug. III. Studies on the mechanism of action. Arzneimittelforschung. 1981;31(9a):1558-65. PubMed PMID: 7197970.