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MedKoo Cat#: 563838 | Name: CJ-1882

Description:

WARNING: This product is for research use only, not for human or veterinary use.

CJ-1882 is a potent and competitive antagonist at the human D3 receptor.

Chemical Structure

CJ-1882
CJ-1882
CAS#NONE

Theoretical Analysis

MedKoo Cat#: 563838

Name: CJ-1882

CAS#: NONE

Chemical Formula: C29H33ClN2O2

Exact Mass: 476.2231

Molecular Weight: 477.05

Elemental Analysis: C, 73.02; H, 6.97; Cl, 7.43; N, 5.87; O, 6.71

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
CJ-1882; CJ-1882; CJ-1882
IUPAC/Chemical Name
Naphthalene-2-carboxylic acid [3-(2-{[2(S)-(4-chloro-phenyl)-1(R)-cyclopropyl]-propyl-amino}-ethyl)-3-hydroxy-cis-cyclobutyl]-amide
InChi Key
KIRKSXHWZHQUBF-YJIPECKFSA-N
InChi Code
InChI=1S/C29H33ClN2O2/c1-2-14-32(27-17-26(27)21-9-11-24(30)12-10-21)15-13-29(34)18-25(19-29)31-28(33)23-8-7-20-5-3-4-6-22(20)16-23/h3-12,16,25-27,34H,2,13-15,17-19H2,1H3,(H,31,33)/t25-,26-,27+,29+/m0/s1
SMILES Code
O=C(N[C@@H]1C[C@@](O)(CCN([C@H]2[C@H](C3=CC=C(Cl)C=C3)C2)CCC)C1)C4=CC5=C(C=C4)C=CC=C5
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 477.05 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Chen J, Levant B, Jiang C, Keck TM, Newman AH, Wang S. Tranylcypromine substituted cis-hydroxycyclobutylnaphthamides as potent and selective dopamine D₃ receptor antagonists. J Med Chem. 2014 Jun 12;57(11):4962-8. doi: 10.1021/jm401798r. Epub 2014 Jun 3. PubMed PMID: 24848155; PubMed Central PMCID: PMC4216217.