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MedKoo Cat#: 461581 | Name: Mazapertine succinate

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Mazapertine succinate is an antipsychotic agent.

Chemical Structure

Mazapertine succinate
Mazapertine succinate
CAS#134208-18-7

Theoretical Analysis

MedKoo Cat#: 461581

Name: Mazapertine succinate

CAS#: 134208-18-7

Chemical Formula: C30H41N3O6

Exact Mass: 539.2995

Molecular Weight: 539.67

Elemental Analysis: C, 66.77; H, 7.66; N, 7.79; O, 17.79

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
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Synonym
Mazapertine succinate; Mazapertine;
IUPAC/Chemical Name
(3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)phenyl)(piperidin-1-yl)methanone succinate
InChi Key
WAHFGTZTVZRLEY-UHFFFAOYSA-N
InChi Code
InChI=1S/C26H35N3O2.C4H6O4/c1-21(2)31-25-12-5-4-11-24(25)28-17-15-27(16-18-28)20-22-9-8-10-23(19-22)26(30)29-13-6-3-7-14-29;5-3(6)1-2-4(7)8/h4-5,8-12,19,21H,3,6-7,13-18,20H2,1-2H3;1-2H2,(H,5,6)(H,7,8)
SMILES Code
O=C(O)CCC(O)=O.O=C(N1CCCCC1)C2=CC=CC(CN3CCN(C4=CC=CC=C4OC(C)C)CC3)=C2
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 539.67 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Ye N, Song Z, Zhang A. Dual ligands targeting dopamine D2 and serotonin 5-HT1A receptors as new antipsychotical or anti-Parkinsonian agents. Curr Med Chem. 2014;21(4):437-57. Review. PubMed PMID: 24164194. 2: Caldwell GW, Wu WN, McKown LA, Diane Gauthier A, Masucci JA, Jones WJ, Leo GC, Reitz AB. Distribution and metabolism of the antipsychotic agent mazapertine succinate in rats. J Pharm Biomed Anal. 2006 May 3;41(2):500-9. Epub 2005 Dec 28. PubMed PMID: 16386397. 3: Wu WN, McKown LA, Takacs AR, Jones WJ, Reitz AB. Biotransformation of the antipsychotic agent, mazapertine, in dog--mass spectral characterization and identification of metabolites. Xenobiotica. 1999 May;29(5):453-66. PubMed PMID: 10379984.