MedKoo Cat#: 592617 | Name: Piprofurol

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Piprofurol is a Calcium channel blocker.

Chemical Structure

Piprofurol
Piprofurol
CAS#40680-87-3

Theoretical Analysis

MedKoo Cat#: 592617

Name: Piprofurol

CAS#: 40680-87-3

Chemical Formula: C26H33NO6

Exact Mass: 455.2308

Molecular Weight: 455.55

Elemental Analysis: C, 68.55; H, 7.30; N, 3.07; O, 21.07

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
No Data
Synonym
Piprofurol; Piprofurolum
IUPAC/Chemical Name
5-Benzofuranmethanol, 4,7-dimethoxy-alpha-(2-(4-hydroxyphenyl)ethyl)-6- (2-(1-piperidinyl)ethoxy)-
InChi Key
LIAPJIQUUKLLDZ-UHFFFAOYSA-N
InChi Code
InChI=1S/C26H33NO6/c1-30-23-20-12-16-32-24(20)26(31-2)25(33-17-15-27-13-4-3-5-14-27)22(23)21(29)11-8-18-6-9-19(28)10-7-18/h6-7,9-10,12,16,21,28-29H,3-5,8,11,13-15,17H2,1-2H3
SMILES Code
OC(CCC1=CC=C(O)C=C1)C2=C(OCCN3CCCCC3)C(OC)=C(OC=C4)C4=C2OC
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 455.55 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Pourrias B, Huerta F, Santamaria R, Bowe C. Calcium blocking properties of piprofurol. Arch Int Pharmacodyn Ther. 1985 Apr;274(2):223-39. PubMed PMID: 4026458. 2: Medvedowsky JL, Barnay C. [Significance of pharmacodynamics tests in the study of sinus node function]. Arch Mal Coeur Vaiss. 1976 Jan;69(1):1-12. French. PubMed PMID: 823883. 3: Barnay C, Medvedowsky JL. [Effect of a depressant drug on the recovery time of the sinus. Attempt of application to the diagnosis of sinus dysfunctions]. Arch Mal Coeur Vaiss. 1977 Sep;70(9):981-6. French. PubMed PMID: 415695.