Tildacerfont | CAS# 1014983-00-6 | CRF antagonist

MedKoo Cat#: 572151 | Name: Tildacerfont

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tildacerfont is a corticotropin releasing factor (CRF) antagonist.

Chemical Structure

Tildacerfont

CAS#1014983-00-6

Theoretical Analysis

MedKoo Cat#: 572151

Name: Tildacerfont

CAS#: 1014983-00-6

Chemical Formula: C20H26ClN5OS

Exact Mass: 419.1547

Molecular Weight: 419.97

Elemental Analysis: C, 57.20; H, 6.24; Cl, 8.44; N, 16.68; O, 3.81; S, 7.63

Price and Availability

Size	Price	Availability
10mg	USD 750.00	2 Weeks
25mg	USD 1,350.00	2 Weeks
50mg	USD 2,450.00	2 Weeks
100mg	USD 3,850.00	2 Weeks

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Related CAS #

No Data

Synonym

Tildacerfont

IUPAC/Chemical Name

4-(4-chloro-5-(2,5-dimethyl-7-(pentan-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl)thiazol-2-yl)morpholine

InChi Key

XVAWSBAQNIXMIO-UHFFFAOYSA-N

InChi Code

InChI=1S/C20H26ClN5OS/c1-5-14(6-2)15-11-12(3)22-19-16(13(4)24-26(15)19)17-18(21)23-20(28-17)25-7-9-27-10-8-25/h11,14H,5-10H2,1-4H3

SMILES Code

CCC(C1=CC(C)=NC2=C(C3=C(Cl)N=C(N4CCOCC4)S3)C(C)=NN12)CC

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.03.00

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 419.97 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Zorrilla EP, Logrip ML, Koob GF. Corticotropin releasing factor: a key role in the neurobiology of addiction. Front Neuroendocrinol. 2014 Apr;35(2):234-44. doi: 10.1016/j.yfrne.2014.01.001. Epub 2014 Jan 20. Review. PubMed PMID: 24456850; PubMed Central PMCID: PMC4213066.