Rad 243 | CAS#103825-20-3 | antiarrhythmic

MedKoo Cat#: 461137 | Name: Rad 243

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Rad 243 is a sodium channel blocker and antiarrhythmic drug.

Chemical Structure

Rad 243

CAS#103825-20-3

Theoretical Analysis

MedKoo Cat#: 461137

Name: Rad 243

CAS#: 103825-20-3

Chemical Formula: C18H30N2O

Exact Mass: 290.2358

Molecular Weight: 290.45

Elemental Analysis: C, 74.44; H, 10.41; N, 9.65; O, 5.51

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

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Related CAS #

No Data

Synonym

Rad 243; Rad-243; Rad243;

IUPAC/Chemical Name

N-(2,6-dimethylphenyl)-2-(heptyl(methyl)amino)acetamide

InChi Key

QVCAEZCAUFJGGS-UHFFFAOYSA-N

InChi Code

InChI=1S/C18H30N2O/c1-5-6-7-8-9-13-20(4)14-17(21)19-18-15(2)11-10-12-16(18)3/h10-12H,5-9,13-14H2,1-4H3,(H,19,21)

SMILES Code

CN(CCCCCCC)CC(Nc1c(C)cccc1C)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.03.00

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 290.45 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Grant AO, Chandra R, Keller C, Carboni M, Starmer CF. Block of wild-type and inactivation-deficient cardiac sodium channels IFM/QQQ stably expressed in mammalian cells. Biophys J. 2000 Dec;79(6):3019-35. PubMed PMID: 11106609; PubMed Central PMCID: PMC1301180. 2: Liu L, Wendt DJ, Grant AO. Relationship between structure and sodium channel blockade by lidocaine and its amino-alkyl derivatives. J Cardiovasc Pharmacol. 1994 Nov;24(5):803-12. PubMed PMID: 7532759.