MedKoo Cat#: 597719 | Name: RX 783030

Description:

WARNING: This product is for research use only, not for human or veterinary use.

RX 783030 is a stabilized enkephalin analog.

Chemical Structure

RX 783030
RX 783030
CAS#72080-55-8

Theoretical Analysis

MedKoo Cat#: 597719

Name: RX 783030

CAS#: 72080-55-8

Chemical Formula: C28H40N6O6

Exact Mass: 556.3009

Molecular Weight: 556.66

Elemental Analysis: C, 60.41; H, 7.24; N, 15.10; O, 17.24

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
RX 783030; RX-783030; RX783030;
IUPAC/Chemical Name
L-Phenylalaninamide, L-tyrosyl-D-alanylglycyl-N-(2-(dimethylamino)ethyl)-N(alpha)-methyl-, N-oxide
InChi Key
RDOMYVAFRDNQBZ-YGOYIFOWSA-N
InChi Code
InChI=1S/C28H40N6O6/c1-19(31-27(38)23(29)16-21-10-12-22(35)13-11-21)26(37)30-18-25(36)34(40)28(39)24(33(4)15-14-32(2)3)17-20-8-6-5-7-9-20/h5-13,19,23-24,34-35H,14-18,29H2,1-4H3,(H,30,37)(H,31,38)/t19-,23+,24+/m1/s1
SMILES Code
O=C([NH+]([O-])C(CNC([C@@H](C)NC([C@H](CC1=CC=C(O)C=C1)N)=O)=O)=O)[C@H](CC2=CC=CC=C2)N(CCN(C)C)C
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 556.66 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Sanger DJ, McCarthy PS. Increased food and water intake produced in rats by opiate receptor agonists. Psychopharmacology (Berl). 1981;74(3):217-20. PubMed PMID: 6791229. 2: Porreca F, LoPresti D, Ward SJ. Opioid agonist affinity in the guinea-pig ileum and mouse vas deferens. Eur J Pharmacol. 1990 Apr 10;179(1-2):129-39. PubMed PMID: 2163849. 3: Smith CF, Waldron C, Brook NA. Opioid receptors in the mouse ileum. Arch Int Pharmacodyn Ther. 1988 Jan-Feb;291:122-31. PubMed PMID: 2835021. 4: Smith CF, Rance MJ. Opiate receptors in the rat vas deferens. Life Sci. 1983;33 Suppl 1:327-30. PubMed PMID: 6319887. 5: Cooper SJ. Effects of opiate agonists and antagonists on fluid intake and saccharin choice in the rat. Neuropharmacology. 1983 Mar;22(3):323-8. PubMed PMID: 6843791. 6: Takemori AE, Portoghese PS. Receptors for opioid peptides in the guinea-pig ileum. J Pharmacol Exp Ther. 1985 Nov;235(2):389-92. PubMed PMID: 2997432.