MedKoo Cat#: 596643 | Name: L 687306

Description:

WARNING: This product is for research use only, not for human or veterinary use.

L 687306 is a partial agonist at muscarinic M1 receptors; a highly competitve antagonist at cardiac M2 receptors and ileal M3 muscarinic receptors.

Chemical Structure

L 687306
L 687306
CAS#139346-23-9

Theoretical Analysis

MedKoo Cat#: 596643

Name: L 687306

CAS#: 139346-23-9

Chemical Formula: C11H15N3O

Exact Mass: 205.1215

Molecular Weight: 205.26

Elemental Analysis: C, 64.37; H, 7.37; N, 20.47; O, 7.79

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
L 687306; L-687306; L687306; L-687,306; L 687,306; L687,306;
IUPAC/Chemical Name
5-(1-azabicyclo[2.2.1]heptan-3-yl)-3-cyclopropyl-1,2,4-oxadiazole
InChi Key
RDPVNJCVSHULSM-UHFFFAOYSA-N
InChi Code
InChI=1S/C11H15N3O/c1-2-7(1)10-12-11(15-13-10)9-6-14-4-3-8(9)5-14/h7-9H,1-6H2
SMILES Code
N1(C2)CC(C3=NC(C4CC4)=NO3)C2CC1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 205.26 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Dawson GR, Iversen SD. The effects of novel cholinesterase inhibitors and selective muscarinic receptor agonists in tests of reference and working memory. Behav Brain Res. 1993 Nov 30;57(2):143-53. PubMed PMID: 8117420. 2: Freedman SB, Patel S, Harley EA, Iversen LL, Baker R, Showell GA, Saunders J, McKnight A, Newberry N, Scholey K, et al. L-687,306: a functionally selective and potent muscarinic M1 receptor agonist. Eur J Pharmacol. 1992 Apr 29;215(1):135-6. PubMed PMID: 1516645.