Tyrphostin 51 | CAS#126433-07-6

MedKoo Cat#: 341202 | Name: Tyrphostin 51

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Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tyrphostin 51 is a potent inhibitor of EGFR (EGF receptor) kinase activity

Chemical Structure

Tyrphostin 51

CAS#126433-07-6

Theoretical Analysis

MedKoo Cat#: 341202

Name: Tyrphostin 51

CAS#: 126433-07-6

Chemical Formula: C13H8N4O3

Exact Mass: 268.0596

Molecular Weight: 268.23

Elemental Analysis: C, 58.21; H, 3.01; N, 20.89; O, 17.89

Price and Availability

Size	Price	Availability	Quantity
5mg	USD 280.00
25mg	USD 750.00

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Related CAS #

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Synonym

Tyrphostin 51; Tyrphostin A 51; Tyrphostin A-51; Tyrphostin A51.

IUPAC/Chemical Name

2-Amino-1,1,3-tricyano-4-(3',4',5'-trihydroxyphenyl)butadiene

InChi Key

JKNOYWVMHPMBEL-UNXLUWIOSA-N

InChi Code

InChI=1S/C13H8N4O3/c14-4-8(12(17)9(5-15)6-16)1-7-2-10(18)13(20)11(19)3-7/h1-3,18-20H,17H2/b8-1+

SMILES Code

c1c(cc(c(c1O)O)O)/C=C(\C#N)/C(=C(C#N)C#N)N

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 268.23 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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L-2-Aminosuberic acid