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MedKoo Cat#: 562056 | Name: TC-I 2014
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

TC-I 2014 is a potent TRPM8 antagonist that exhibits antiallodynic properties in pain models.

Chemical Structure

TC-I 2014
TC-I 2014
CAS#1221349-53-6

Theoretical Analysis

MedKoo Cat#: 562056

Name: TC-I 2014

CAS#: 1221349-53-6

Chemical Formula: C23H19F6N3O

Exact Mass: 467.1432

Molecular Weight: 467.41

Elemental Analysis: C, 59.10; H, 4.10; F, 24.39; N, 8.99; O, 3.42

Price and Availability

Size Price Availability Quantity
50mg USD 850.00 2 Weeks
100mg USD 1,450.00 2 Weeks
200mg USD 2,150.00 2 Weeks
500mg USD 3,250.00 2 Weeks
1g USD 4,650.00 2 Weeks
2g USD 6,850.00 2 Weeks
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Related CAS #
No Data
Synonym
TC-I 2014; TC I 2014; TCI 2014;
IUPAC/Chemical Name
3-[7-(Trifluoromethyl)-5-[2-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl]-1-oxa-2-azaspiro[4.5]dec-2-ene
InChi Key
VSMFCZZEKTVDHM-UHFFFAOYSA-N
InChi Code
InChI=1S/C23H19F6N3O/c24-22(25,26)15-7-3-2-6-14(15)13-10-16(23(27,28)29)19-17(11-13)30-20(31-19)18-12-21(33-32-18)8-4-1-5-9-21/h2-3,6-7,10-11H,1,4-5,8-9,12H2,(H,30,31)
SMILES Code
FC(C1=CC=CC=C1C2=CC(C(F)(F)F)=C3C(N=C(C4=NOC5(CCCCC5)C4)N3)=C2)(F)F
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 467.41 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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