KUN75125 is a phosphodiesterase-4 (PDE4) allosteric modulator with IC50 values of 8 and 130 nM against human and mouse PDE4D, respectivel. It may help reverse scopolamine-induced cognitive impairment.
MedKoo Cat#: 571494
Name: KUN75125
CAS#: 1606975-12-5
Chemical Formula: C19H14ClF3N4O
Exact Mass: 406.0808
Molecular Weight: 406.79
Elemental Analysis: C, 56.10; H, 3.47; Cl, 8.71; F, 14.01; N, 13.77; O, 3.93
The following data is based on the product molecular weight 406.79 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
