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MedKoo Cat#: 527072 | Name: 4-Amino-PPHT Hydrobromide

Description:

WARNING: This product is for research use only, not for human or veterinary use.

4-Amino-PPHT Hydrobromide is a precursor for fluorescent labeled Dopamine D2 receptors (D2R) agonist.

Chemical Structure

4-Amino-PPHT Hydrobromide
4-Amino-PPHT Hydrobromide
CAS#129298-03-9

Theoretical Analysis

MedKoo Cat#: 527072

Name: 4-Amino-PPHT Hydrobromide

CAS#: 129298-03-9

Chemical Formula: C21H29BrN2O

Exact Mass: 404.1463

Molecular Weight: 405.38

Elemental Analysis: C, 62.22; H, 7.21; Br, 19.71; N, 6.91; O, 3.95

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
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Synonym
4-Amino-PPHT Hydrobromide
IUPAC/Chemical Name
6-[[2-(4-Aminophenyl)ethyl]propylamino]-5,6,7,8-tetrahydro-1-naphthalenol hydrobromide
InChi Key
JLEJPNRRWHBLOH-UHFFFAOYSA-N
InChi Code
InChI=1S/C21H28N2O.BrH/c1-2-13-23(14-12-16-6-8-18(22)9-7-16)19-10-11-20-17(15-19)4-3-5-21(20)24;/h3-9,19,24H,2,10-15,22H2,1H3;1H
SMILES Code
OC1=C2CCC(N(CCC3=CC=C(N)C=C3)CCC)CC2=CC=C1.[H]Br
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 405.38 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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Detection of scopolamine and atropine in organic buckwheat (Fagopyron esculentum L.) products by UHPLC-MS/MS. Food Chem. 2018 Jan 15;239:141-147. doi: 10.1016/j.foodchem.2017.06.028. Epub 2017 Jun 23. PubMed PMID: 28873551. 11: Ponzoni L, Braida D, Bondiolotti G, Sala M. The Non-Peptide Arginine-Vasopressin v(1a) Selective Receptor Antagonist, SR49059, Blocks the Rewarding, Prosocial, and Anxiolytic Effects of 3,4-Methylenedioxymethamphetamine and Its Derivatives in Zebra Fish. Front Psychiatry. 2017 Aug 14;8:146. doi: 10.3389/fpsyt.2017.00146. eCollection 2017. PubMed PMID: 28855876; PubMed Central PMCID: PMC5557732. 12: Lin Q, Jia Z, Xu X, Xu S, Han T, Gao Y, Zhang Y, Zhang H, Liu H, Li J, Li X. Sub-chronic toxicity study of arecae semen aqueous extract in Wistar rats. J Ethnopharmacol. 2017 Aug 25. pii: S0378-8741(16)32236-X. doi: 10.1016/j.jep.2017.08.031. 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