MedKoo Cat#: 526413 | Name: RG-102240

Description:

WARNING: This product is for research use only, not for human or veterinary use.

RG-102240 is a gene switch ligand as a transcription inducer for use in induceable gene expression systems.

Chemical Structure

RG-102240
RG-102240
CAS#162326-49-0

Theoretical Analysis

MedKoo Cat#: 526413

Name: RG-102240

CAS#: 162326-49-0

Chemical Formula: C23H30N2O3

Exact Mass: 382.2256

Molecular Weight: 382.50

Elemental Analysis: C, 72.22; H, 7.91; N, 7.32; O, 12.55

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
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Synonym
RG-102240; RG 102240; RG102240
IUPAC/Chemical Name
2-Ethyl-3-methoxybenzoic acid 2-(3,5-dimethylbenzoyl)-2-(1,1-dimethylethyl)hydrazide
InChi Key
QYYXITIZXRMPSZ-UHFFFAOYSA-N
InChi Code
InChI=1S/C23H30N2O3/c1-8-18-19(10-9-11-20(18)28-7)21(26)24-25(23(4,5)6)22(27)17-13-15(2)12-16(3)14-17/h9-14H,8H2,1-7H3,(H,24,26)
SMILES Code
O=C(NN(C(C1=CC(C)=CC(C)=C1)=O)C(C)(C)C)C2=CC=CC(OC)=C2CC
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 382.50 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Bitra K, Palli SR. Interaction of proteins involved in ecdysone and juvenile hormone signal transduction. Arch Insect Biochem Physiol. 2009 Feb;70(2):90-105. doi: 10.1002/arch.20281. PubMed PMID: 18980211. 2: Panguluri SK, Li B, Hormann RE, Palli SR. Effect of ecdysone receptor gene switch ligands on endogenous gene expression in 293 cells. FEBS J. 2007 Nov;274(21):5669-89. Epub 2007 Oct 8. PubMed PMID: 17922837. 3: Kumar MB, Fujimoto T, Potter DW, Deng Q, Palli SR. A single point mutation in ecdysone receptor leads to increased ligand specificity: implications for gene switch applications. Proc Natl Acad Sci U S A. 2002 Nov 12;99(23):14710-5. Epub 2002 Oct 31. PubMed PMID: 12411578; PubMed Central PMCID: PMC137484.