CAY10574, also known as Cdk9 Inhibitor II, is a potent, selective inhibitor of Cdk9 in vitro with an IC50 value of 0.35 µM. It is also a competitive inhibitor of Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 and 20 µM, respectively.
MedKoo Cat#: 407495
Name: CAY10574
CAS#: 140651-18-9
Chemical Formula: C9H10N6O
Exact Mass: 218.0916
Molecular Weight: 218.22
Elemental Analysis: C, 49.54; H, 4.62; N, 38.51; O, 7.33
The following data is based on the product molecular weight 218.22 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
