WAY200070 | CAS#440122-66-7 | ERβ Receptor Agonist

MedKoo Cat#: 532961 | Name: WAY200070

Description:

WARNING: This product is for research use only, not for human or veterinary use.

WAY200070 is a selective ERβ receptor agonist that displays 68-fold selectivity over ERα (EC50 values are 2 and 155 nM for ERβ and ERα respectively). WAY200070 displays antianxiolytic and antidepressive effects in vivo.

Chemical Structure

WAY200070

CAS#440122-66-7

Theoretical Analysis

MedKoo Cat#: 532961

Name: WAY200070

CAS#: 440122-66-7

Chemical Formula: C13H8BrNO3

Exact Mass: 304.9688

Molecular Weight: 306.12

Elemental Analysis: C, 51.01; H, 2.63; Br, 26.10; N, 4.58; O, 15.68

Price and Availability

Size	Price	Availability
50mg	USD 450.00	2 Weeks
100mg	USD 750.00	2 Weeks
200mg	USD 1,350.00	2 Weeks
500mg	USD 2,850.00	2 Weeks
1g	USD 4,250.00	2 Weeks
2g	USD 7,450.00	2 Weeks

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Related CAS #

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Synonym

WAY200070; WAY 200070; WAY-200070

IUPAC/Chemical Name

4-(7-bromo-5-hydroxy-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,5-dien-1-one

InChi Key

IVFWABSHZFOMIG-UHFFFAOYSA-N

InChi Code

InChI=1S/C13H8BrNO3/c14-10-5-9(17)6-11-12(10)18-13(15-11)7-1-3-8(16)4-2-7/h1-6,15,17H

SMILES Code

O=C1C=C/C(C=C1)=C2OC3=C(Br)C=C(O)C=C3N/2

Appearance

White to beige solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 306.12 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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