TP003 is a functionally selective GABAA receptor (α3 subtype) partial agonist. TP003 exhibits affinity for the benzodiazepine binding site on human GABAA receptors. It potentiates the GABA (α3 subtype) response selectively with high efficacy.
MedKoo Cat#: 532821
Name: TP003
CAS#: 628690-75-5
Chemical Formula: C23H16F3N3O
Exact Mass: 407.1245
Molecular Weight: 407.40
Elemental Analysis: C, 67.81; H, 3.96; F, 13.99; N, 10.31; O, 3.93
The following data is based on the product molecular weight 407.40 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
