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MedKoo Cat#: 531781 | Name: FG-5893

Description:

WARNING: This product is for research use only, not for human or veterinary use.

FG-5893 is a novel 5-HT1A agonist/5-HT2 antagonist. FG-5893 is a potential anxiolytic drug.

Chemical Structure

FG-5893
FG-5893
CAS#150527-23-4

Theoretical Analysis

MedKoo Cat#: 531781

Name: FG-5893

CAS#: 150527-23-4

Chemical Formula: C27H29F2N3O2

Exact Mass: 465.2228

Molecular Weight: 465.54

Elemental Analysis: C, 69.66; H, 6.28; F, 8.16; N, 9.03; O, 6.87

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
FG-5893; FG 5893; FG5893.
IUPAC/Chemical Name
methyl 2-[4-[4,4-bis(4-fluorophenyl)butyl]piperazin-1-yl]pyridine-3-carboxylate
InChi Key
NDCPNKXUTJGQQC-UHFFFAOYSA-N
InChi Code
InChI=1S/C27H29F2N3O2/c1-34-27(33)25-4-2-14-30-26(25)32-18-16-31(17-19-32)15-3-5-24(20-6-10-22(28)11-7-20)21-8-12-23(29)13-9-21/h2,4,6-14,24H,3,5,15-19H2,1H3
SMILES Code
O=C(C1=CC=CN=C1N2CCN(CCCC(C3=CC=C(F)C=C3)C4=CC=C(F)C=C4)CC2)OC
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 465.54 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Lankford MF, Björk AK, Myers RD. Differential efficacy of serotonergic drugs FG5974, FG5893, and amperozide in reducing alcohol drinking in P rats. Alcohol. 1996 Jul-Aug;13(4):399-404. PubMed PMID: 8836330. 2: Long TA, Kalmus GW, Björk A, Myers RD. Alcohol intake in high alcohol drinking (HAD) rats is suppressed by FG5865, a novel 5-HT1A agonist/5-HT2 antagonist. Pharmacol Biochem Behav. 1996 Jan;53(1):33-40. PubMed PMID: 8848457.