MedKoo Cat#: 531309 | Name: SU 4942
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

SU-4942 is a tyrosine kinase signal signal modulator. SU-4942 inhibits VEGF- and endothelial cell growth factor (ECGF)-induced mitogenesis in endothelial cells.

Chemical Structure

SU 4942
SU 4942
CAS#76086-99-2

Theoretical Analysis

MedKoo Cat#: 531309

Name: SU 4942

CAS#: 76086-99-2

Chemical Formula: C15H10BrNO

Exact Mass: 298.9946

Molecular Weight: 300.16

Elemental Analysis: C, 60.02; H, 3.36; Br, 26.62; N, 4.67; O, 5.33

Price and Availability

Size Price Availability Quantity
100mg USD 650.00 2 weeks
200mg USD 950.00 2 weeks
500mg USD 1,650.00 2 weeks
1g USD 2,650.00 2 weeks
2g USD 3,850.00 2 weeks
5g USD 5,750.00 2 weeks
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Related CAS #
No Data
Synonym
SU 4942; SU-4942; SU4942.
IUPAC/Chemical Name
3-(4-Bromobenzylidene)-1,3-dihydroindol-2-one
InChi Key
INAOSTJXLBNFMV-LCYFTJDESA-N
InChi Code
InChI=1S/C15H10BrNO/c16-11-7-5-10(6-8-11)9-13-12-3-1-2-4-14(12)17-15(13)18/h1-9H,(H,17,18)/b13-9-
SMILES Code
O=C1NC2=C(C=CC=C2)/C1=C/C3=CC=C(Br)C=C3
Appearance
Yellow solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info
Product Data
Biological target:
SU 4942 is a bioactive chemical.
In vitro activity:
To be determined
In vivo activity:
To be determined
Solvent mg/mL mM
Solubility
DMF 30.0 99.95
DMSO 30.0 99.95
Ethanol 1.0 3.33
Note: There can be variations in solubility for the same chemical from different vendors or different batches from the same vendor. The following factors can affect the solubility of the same chemical: solvent used for crystallization, residual solvent content, polymorphism, salt versus free form, degree of hydration, solvent temperature. Please use the solubility data as a reference only. Warming and sonication will facilitate dissolving. Still have questions? Please contact our Technical Support scientists.

Preparing Stock Solutions

The following data is based on the product molecular weight 300.16 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
To be determined
In vitro protocol:
To be determined
In vivo protocol:
To be determined
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