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MedKoo Cat#: 525911 | Name: Peliglitazar

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Peliglitazar is a dual α/γ peroxisome proliferator-activated receptor activator.

Chemical Structure

Peliglitazar
Peliglitazar
CAS#331744-64-0

Theoretical Analysis

MedKoo Cat#: 525911

Name: Peliglitazar

CAS#: 331744-64-0

Chemical Formula: C30H30N2O7

Exact Mass: 530.2053

Molecular Weight: 530.58

Elemental Analysis: C, 67.91; H, 5.70; N, 5.28; O, 21.11

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Peliglitazar; BMS 426707-01; BMS-426707-1; BMS 42670701.
IUPAC/Chemical Name
Glycine, N-((4-methoxyphenoxy)carbonyl)-N-((1S)-1-(4-(2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy)phenyl)ethyl)-
InChi Key
CUADMYMMZWFUCY-FQEVSTJZSA-N
InChi Code
InChI=1S/C30H30N2O7/c1-20(32(19-28(33)34)30(35)39-26-15-13-24(36-3)14-16-26)22-9-11-25(12-10-22)37-18-17-27-21(2)38-29(31-27)23-7-5-4-6-8-23/h4-16,20H,17-19H2,1-3H3,(H,33,34)/t20-/m0/s1
SMILES Code
O=C(O)CN(C(OC1=CC=C(OC)C=C1)=O)[C@H](C2=CC=C(OCCC3=C(C)OC(C4=CC=CC=C4)=N3)C=C2)C
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 530.58 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Wang L, Munsick C, Chen S, Bonacorsi S, Cheng PT, Humphreys WG, Zhang D. Metabolism and disposition of 14C-labeled peliglitazar in humans. Drug Metab Dispos. 2011 Feb;39(2):228-38. doi: 10.1124/dmd.110.035089. Epub 2010 Oct 26. PubMed PMID: 20978103. 2: Zhang D, Raghavan N, Wang L, Xue Y, Obermeier M, Chen S, Tao S, Zhang H, Cheng PT, Li W, Ramanathan R, Yang Z, Humphreys WG. Plasma stability-dependent circulation of acyl glucuronide metabolites in humans: how circulating metabolite profiles of muraglitazar and peliglitazar can lead to misleading risk assessment. Drug Metab Dispos. 2011 Jan;39(1):123-31. doi: 10.1124/dmd.110.035048. Epub 2010 Sep 28. PubMed PMID: 20876787.