1: Sammons MF, Lee EC. Recent progress in the development of small-molecule
glucagon receptor antagonists. Bioorg Med Chem Lett. 2015 Oct 1;25(19):4057-64.
doi: 10.1016/j.bmcl.2015.07.092. Review. PubMed PMID: 26271588.
1. Methods of treating diabetes by administering a glucagon receptor antagonist in combination with a cholesterol absorption inhibitor
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By Guan, Hong-Ping; Castro-Perez, Jose M.; Davis, Harry R.; Engel, Samuel S.; Johns, Douglas G.; Lin, Songnian; Previs, Steven F.; Roddy, Thomas P.; Wang, Liangsu; Wang, Sheng-Ping; et al
From PCT Int. Appl. (2014), WO 2014093189 A1 20140619. | Language: English, Database: CAPLUS
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2. The design and synthesis of a potent glucagon receptor antagonist with favorable physicochemical and pharmacokinetic properties as a candidate for the treatment of type 2 diabetes mellitus
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By Guzman-Perez, Angel; Pfefferkorn, Jeffrey A.; Lee, Esther C. Y.; Stevens, Benjamin D.; Aspnes, Gary E.; Bian, Jianwei; Didiuk, Mary T.; Filipski, Kevin J.; Moore, Dianna; Perreault, Christian; et al
From Bioorganic & Medicinal Chemistry Letters (2013), 23(10), 3051-3058. | Language: English, Database: CAPLUS
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3. Asymmetric Synthesis of a Glucagon Receptor Antagonist via Friedel-Crafts Alkylation of Indole with Chiral α-Phenyl Benzyl Cation
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By Chung, John Y. L.; Steinhuebel, Dietrich; Krska, Shane W.; Hartner, Fred W.; Cai, Chaoxian; Rosen, Jonathan; Mancheno, Danny E.; Pei, Tao; DiMichele, Lisa; Ball, Richard G.; et al
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4. A novel series of glucagon receptor antagonists with reduced molecular weight and lipophilicity
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From Bioorganic & Medicinal Chemistry Letters (2012), 22(1), 415-420. | Language: English, Database: CAPLUS
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5. Glucagon receptor antagonist compounds, compositions containing such compounds and methods of use
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From PCT Int. Appl. (2010), WO 2010098994 A1 20100902. | Language: English, Database: CAPLUS
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6. Preparation of indole β-alanine derivatives as glucagon receptor antagonist
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By Stelmach, John E.; Parmee, Emma R.; Tata, James R.; Rosauer, Keith G.; Kim, Ronald M.; Bittner, Amy R.; Chang, Jiang; Sinz, Christopher Joseph
From U.S. (2010), US 7687534 B2 20100330. | Language: English, Database: CAPLUS
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7. Preparation of 1,2-diphenylethane compounds as glucagon receptor antagonist for diabetes treatment
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From PCT Int. Appl. (2010), WO 2010030722 A1 20100318. | Language: English, Database: CAPLUS
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8. Preparation of indole β-alanine derivatives as glucagon receptor antagonist
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By Stelmach, John E.; Parmee, Emma R.; Tata, James R.; Rosauer, Keith G.; Kim, Ronald M.; Bittner, Amy R.; Chang, Jiang; Sinz, Christopher Joseph
From PCT Int. Appl. (2008), WO 2008042223 A1 20080410. | Language: English, Database: CAPLUS
