Pitolisant, also known as Tiprolisant, BF2649 and Ciproxidine, is a histamine receptor inverse agonist/antagonist selective for the H3 subtype. It has stimulant and nootropic effects and may have several medical applications such as treatment of narcolepsy
Qu, Chang; Liang, Chuang; Lu, Ying-xiang; Yang, Gui-qiu; Gong, Ping Zhongguo Yaowu Huaxue Zazhi. Synthesis of pitolisant as a histamine H3 receptor antagonist/invers Zhongguo Yaowu Huaxue Zazhi. Volume 23. Issue 2. Pages 111-114. Journal. (2013).
